Structural basis for the function of DCN-1 in protein Neddylation

J Biol Chem. 2007 Aug 24;282(34):24490-4. doi: 10.1074/jbc.C700038200. Epub 2007 Jun 26.

Abstract

Covalent modification by Nedd8 (neddylation) stimulates the ubiquitin-protein isopeptide ligase (E3) activities of Cullins. DCN-1, an evolutionarily conserved protein, promotes neddylation of Cullins in vivo, binds directly to Nedd8, and associates with Cdc53 in the budding yeast Saccharomyces cerevisiae. The 1.9A resolution structure of yeast DCN-1 shows that the region encompassing residues 66-269 has a rectangular parallelepiped-like all alpha-helical structures, consisting of an EF-hand motif N-terminal domain and a closely juxtaposed C-terminal domain with six alpha-helices. The EF-hand motif structure is highly similar to that of the c-Cbl ubiquitin E3 ligase. We also demonstrate that DCN-1 directly binds to Rbx-1, a factor important for protein neddylation. The structural and biochemical results are consistent with the role of DCN-1 as a scaffold protein in a multisubunit neddylation E3 ligase complex.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Motifs
  • Amino Acid Sequence
  • Animals
  • Cell Cycle Proteins / metabolism
  • Conserved Sequence
  • Cullin Proteins / metabolism
  • Evolution, Molecular
  • Humans
  • Molecular Conformation
  • Molecular Sequence Data
  • NEDD8 Protein
  • Protein Structure, Tertiary
  • Saccharomyces cerevisiae / metabolism
  • Saccharomyces cerevisiae Proteins / chemistry
  • Saccharomyces cerevisiae Proteins / metabolism
  • Saccharomyces cerevisiae Proteins / physiology*
  • Sequence Homology, Amino Acid
  • Ubiquitin-Protein Ligases / metabolism
  • Ubiquitins / metabolism*

Substances

  • Cdc53 protein, S cerevisiae
  • Cell Cycle Proteins
  • Cullin Proteins
  • Dcn1 protein, S cerevisiae
  • NEDD8 Protein
  • NEDD8 protein, human
  • Saccharomyces cerevisiae Proteins
  • Ubiquitins
  • Ubiquitin-Protein Ligases

Associated data

  • PDB/21S9