Kruppel-like factor 5 modulates p53-independent apoptosis through Pim1 survival kinase in cancer cells

Oncogene. 2008 Jan 3;27(1):1-8. doi: 10.1038/sj.onc.1210625. Epub 2007 Jul 2.

Abstract

Although Kruppel-like factor 5 (KLF5) is a transcription factor that has been implicated in pathways critical to carcinogenesis, controversy persists as to whether it functions as a tumor suppressor or as an oncogene. Here, we describe a novel role for KLF5 in a p53-independent apoptotic pathway. Using RNA-interference technology, we show that cells deficient in KLF5 have increased sensitivity to DNA damage, regardless of p53 status. Both p53 and p53-dependent factors are unaffected by KLF5 depletion. Instead, the apoptotic phenotype consequent to damage is associated with reduced bad phosphorylation, and downregulation of Pim1. Consistently, transfection of wild-type Pim1 is sufficient to rescue this phenotype. Previous data have shown a number of putative Sp1-binding consensus sequences on the Pim1 promoter. Remarkably, chromatin immunoprecipitation studies show that KLF5 binds to the Pim1 promoter, and that binding increases soon after damage. These results identify a novel, p53-independent apoptotic pathway through which KLF5 functions in response to DNA damage. Therapeutic deregulation of this pathway could be used to modulate chemosensitivity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis / genetics
  • Apoptosis / physiology*
  • Apoptosis Regulatory Proteins / deficiency
  • Apoptosis Regulatory Proteins / genetics
  • Apoptosis Regulatory Proteins / physiology*
  • Cell Survival / genetics
  • Cell Survival / physiology
  • DNA Damage / genetics
  • HCT116 Cells
  • Humans
  • Kruppel-Like Transcription Factors / genetics
  • Kruppel-Like Transcription Factors / metabolism
  • Kruppel-Like Transcription Factors / physiology*
  • Phosphorylation
  • Protein Binding / genetics
  • Proto-Oncogene Proteins c-pim-1 / biosynthesis
  • Proto-Oncogene Proteins c-pim-1 / genetics
  • Proto-Oncogene Proteins c-pim-1 / physiology*
  • Signal Transduction / genetics
  • Transfection
  • Tumor Suppressor Protein p53 / deficiency
  • Tumor Suppressor Protein p53 / genetics
  • Tumor Suppressor Protein p53 / physiology*
  • bcl-Associated Death Protein / metabolism

Substances

  • Apoptosis Regulatory Proteins
  • KLF5 protein, human
  • Kruppel-Like Transcription Factors
  • Tumor Suppressor Protein p53
  • bcl-Associated Death Protein
  • PIM1 protein, human
  • Proto-Oncogene Proteins c-pim-1