Brn3 transcription factors control terminal osteoclastogenesis

J Cell Biochem. 2007 Sep 1;102(1):1-12. doi: 10.1002/jcb.21257.

Abstract

Osteoclastic bone resorption is a central mechanism in skeletal development, remodeling and pathology. RANKL is a mandatory factor controlling osteoclastogenesis; however, the underlying signaling pathways are only partially characterized. Using a screening array for the investigation of differential transcription factor activation, we identified activation of the Brn3 transcription factor family as a downstream event of RANKL signaling during terminal osteoclastogenesis. RANKL stimulation induces expression of Brn3a and b and maximal transcriptional activity of Brn3 family members concurrent with osteoclastic giant cell formation. Immunohistochemical analysis revealed both nuclear and cytoplasmic localization of Brn3a and b in mature osteoclasts. Functional inhibition of Brn3 transcription factors resulted in inhibition of pre-osteoclast fusion and reduction in bone resorbing activity of mature osteoclasts. Furthermore, we identified synaptotagmin-1, a regulator of membrane and vesicular fusion, as downstream target of Brn3 with a role in osteoclast function. We conclude that Brn-3 represents a novel molecular differentiation factor that controls osteoclast maturation and function, suggesting an important role in bone metabolism.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Base Sequence
  • Bone Resorption
  • Cell Differentiation
  • Cells, Cultured
  • Consensus Sequence
  • Homeodomain Proteins / antagonists & inhibitors
  • Homeodomain Proteins / metabolism
  • Homeodomain Proteins / physiology*
  • Mice
  • Mice, Inbred BALB C
  • Oligonucleotides / chemistry
  • Osteoclasts / cytology
  • Osteoclasts / metabolism
  • Osteoclasts / physiology*
  • Synaptotagmin I / physiology
  • Transcription Factor Brn-3A / antagonists & inhibitors
  • Transcription Factor Brn-3A / metabolism
  • Transcription Factor Brn-3A / physiology*
  • Transcription Factor Brn-3B / antagonists & inhibitors
  • Transcription Factor Brn-3B / metabolism
  • Transcription Factor Brn-3B / physiology*
  • Transcriptional Activation

Substances

  • Homeodomain Proteins
  • Oligonucleotides
  • Pou4f1 protein, mouse
  • Pou4f2 protein, mouse
  • Synaptotagmin I
  • Syt1 protein, mouse
  • Transcription Factor Brn-3A
  • Transcription Factor Brn-3B