Target assessment for antiparasitic drug discovery

Trends Parasitol. 2007 Dec;23(12):589-95. doi: 10.1016/j.pt.2007.08.019. Epub 2007 Oct 24.

Abstract

Drug discovery is a high-risk, expensive and lengthy process taking at least 12 years and costing upwards of US$500 million per drug to reach the clinic. For neglected diseases, the drug discovery process is driven by medical need and guided by pre-defined target product profiles. Assessment and prioritisation of the most promising targets for entry into screening programmes is crucial for maximising the chances of success. Here, we describe criteria used in our drug discovery unit for target assessment and introduce the 'traffic-light' system as a prioritisation and management tool. We hope this brief review will stimulate basic scientists to acquire additional information necessary for drug discovery.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Antiparasitic Agents / pharmacology*
  • Chemistry, Pharmaceutical
  • Drug Design*
  • Drug Evaluation, Preclinical / economics
  • Drug Evaluation, Preclinical / methods
  • Drug Industry / economics*
  • Humans
  • Parasites / drug effects*
  • Parasitic Diseases / drug therapy*
  • Parasitic Sensitivity Tests
  • Pharmacogenetics
  • Research Design
  • Treatment Outcome

Substances

  • Antiparasitic Agents