Synthesis and structure-immunosuppressive activity relationships of bakuchiol and its derivatives

Bioorg Med Chem. 2008 Mar 1;16(5):2403-11. doi: 10.1016/j.bmc.2007.11.054. Epub 2007 Nov 28.

Abstract

A series of derivatives of bakuchiol were synthesized and tested in vitro for their cytotoxicity, and inhibition of T cell proliferation and B cell proliferation. The data obtained provided preliminary structure-activity relationships of the compounds as immunosuppressive activity.

MeSH terms

  • Animals
  • Cell Proliferation / drug effects
  • Cells, Cultured
  • Concanavalin A / pharmacology
  • Cytoprotection / drug effects
  • Immunosuppressive Agents / chemical synthesis*
  • Immunosuppressive Agents / chemistry
  • Immunosuppressive Agents / pharmacology*
  • Lipopolysaccharides / pharmacology
  • Lymphocytes / cytology
  • Lymphocytes / drug effects
  • Mice
  • Molecular Structure
  • Phenols / chemical synthesis*
  • Phenols / chemistry
  • Phenols / pharmacology*
  • Structure-Activity Relationship

Substances

  • Immunosuppressive Agents
  • Lipopolysaccharides
  • Phenols
  • Concanavalin A
  • bakuchiol