Apoptosis is not the major death mechanism induced by celecoxib on rheumatoid arthritis synovial fibroblasts

Arthritis Res Ther. 2007;9(6):R128. doi: 10.1186/ar2342.

Abstract

Synovial hyperplasia in rheumatoid arthritis (RA) has been associated with apoptosis deficiency of RA fibroblast-like synoviocytes (FLSs). Celecoxib is a non-steroidal anti-inflammatory drug that has been demonstrated to induce apoptosis in some cellular systems. We have therefore examined the dose- and time-dependent effects of celecoxib on RA FLS viability. Treatment of RA FLSs with celecoxib for 24 hours reduced their viability in a dose-dependent manner. Analysis of celecoxib-treated RA FLSs for their content of apoptotic and necrotic cells by Annexin V staining and TO-PRO-3 uptake displayed only few apoptotic cells. Caspase 3, a key mediator of apoptosis, was not activated in celecoxib-treated RA FLSs, and the presence of specific caspase 3 or pan-caspase inhibitors did not affect celecoxib-induced cell death. Moreover, we could not detect other signs of apoptosis, such as cleavage of poly(ADP-ribose) polymerase, caspase 8 or 9, or DNA fragmentation. We therefore conclude that apoptosis is not the major death pathway in celecoxib-treated RA FLSs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Annexin A5 / metabolism
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Apoptosis / drug effects
  • Arthritis, Rheumatoid / drug therapy*
  • Arthritis, Rheumatoid / metabolism
  • Arthritis, Rheumatoid / pathology
  • Caspase 3 / metabolism
  • Celecoxib
  • Cell Death / drug effects
  • Cell Proliferation / drug effects
  • Cells, Cultured
  • Cyclooxygenase Inhibitors / pharmacology*
  • Fibroblasts / drug effects
  • Fibroblasts / pathology
  • Humans
  • Pyrazoles / pharmacology*
  • Staurosporine / pharmacology
  • Sulfonamides / pharmacology*
  • Synovial Membrane / drug effects*
  • Synovial Membrane / pathology
  • TNF-Related Apoptosis-Inducing Ligand / pharmacology

Substances

  • Annexin A5
  • Anti-Inflammatory Agents, Non-Steroidal
  • Cyclooxygenase Inhibitors
  • Pyrazoles
  • Sulfonamides
  • TNF-Related Apoptosis-Inducing Ligand
  • TNFSF10 protein, human
  • CASP3 protein, human
  • Caspase 3
  • Staurosporine
  • Celecoxib