Controlled release of hydrocortisone acetate from dermal bases

Eur J Drug Metab Pharmacokinet. 1991:Spec No 3:466-72.

Abstract

The effect of the complexation with beta-cyclodextrin, hydroxypropyl beta-cyclodextrin and polyvinylpyrrolidone on the diffusion kinetics of hydrocortisone acetate through a non porous lipidic membrane was analyzed starting from different dermal bases: a Carbopol gel and lanovaseline. A constant diffusive gradient was achieved; this suggests that the complexation equilibrium controls the diffusable form, according to its stability constant. The following sequence was observed for the cumulative amount diffused: hydrocortisone acetate greater than hydrocortisone acetate/polyvinylpyrrolidone greater than hydrocortisone acetate/hydroxypropyl beta-cyclodextrin greater than hydrocortisone acetate/beta-cyclodextrin. Such behaviour was analyzed in terms of the main physical chemical parameters of the systems examined.

MeSH terms

  • Acrylic Resins
  • Administration, Topical
  • Chemical Phenomena
  • Chemistry, Physical
  • Cyclodextrins / administration & dosage
  • Diffusion
  • Hydrocortisone / administration & dosage
  • Hydrocortisone / analogs & derivatives*
  • Hydrocortisone / pharmacokinetics
  • Membranes, Artificial
  • Polyvinyls / administration & dosage
  • Povidone / administration & dosage
  • Silicone Elastomers
  • beta-Cyclodextrins*

Substances

  • Acrylic Resins
  • Cyclodextrins
  • Membranes, Artificial
  • Polyvinyls
  • Silicone Elastomers
  • beta-Cyclodextrins
  • carboxypolymethylene
  • hydrocortisone acetate
  • Povidone
  • betadex
  • Hydrocortisone