[3H]MK-801 binding to forebrain of E1 (epileptic) and non-epileptic strains of mice

Epilepsy Res. 1991 Apr;8(3):220-5. doi: 10.1016/0920-1211(91)90067-p.

Abstract

The El mouse is an animal model with genetically determined epilepsy. To elucidate the mechanism of convulsive seizures in El mice, the effects of L-glutamate and glycine on the binding of (+)[3H]MK-801 were studied in well-washed membranes from forebrains of ddY, BALB/c and El (stimulated and non-stimulated) mice. There were no significant differences in affinity (Kd) or density (Bmax) among the 4 groups of mice under basal conditions. Incubation in the presence of L-glutamate and/or glycine led to an increase in apparent density, but not in affinity. No significant change was observed in either Kd, Bmax, or the percentage increase in (+)[3H]MK-801 binding amount the 4 groups in the presence of L-glutamate and/or glycine. These results suggest that the seizure susceptibility of El mice cannot be explained by changes in affinity or density of the NMDA receptor/channel complex.

MeSH terms

  • Animals
  • Brain / drug effects
  • Brain / metabolism*
  • Dizocilpine Maleate / metabolism*
  • Epilepsy / metabolism*
  • Glutamates / pharmacology
  • Glycine / pharmacology
  • Kinetics
  • Mice
  • Radioligand Assay
  • Receptors, N-Methyl-D-Aspartate / metabolism

Substances

  • Glutamates
  • Receptors, N-Methyl-D-Aspartate
  • Dizocilpine Maleate
  • Glycine