The effect of lead on calcium release activated calcium influx in primary cultures of human osteoblast-like cells

Arch Pharm Res. 2008 Feb;31(2):188-94. doi: 10.1007/s12272-001-1140-3.

Abstract

To further understand the significance of bone as a target tissues of lead toxicity, as well as a reservoir of systemic lead, it is necessary to define the effect of lead on the calcium release activated calcium influx (CRACI) in primary cultures of human osteoblast-like cells (OLC). Pb2+ inhibited the immediate CRACI dose-dependent manner. Influx of Pb2+ into human OLC was increased dose-dependent manner. The present study demonstrates that the interference of Pb2+ with CRACI of human OLC is at least twofold: (1) the initiation of CRACI, i.e., the measurable influx of Ca2+ upon Ca2+ readdition, is partially inhibited by Pb2+ and (2) the influx of Pb2+ was enhanced after CRACI had been induced.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calcimycin / pharmacology
  • Calcium / metabolism*
  • Calcium Channels / metabolism
  • Cells, Cultured
  • Data Interpretation, Statistical
  • Enzyme Inhibitors / pharmacology
  • Humans
  • Indicators and Reagents
  • Ionophores / pharmacology
  • Lead / pharmacology*
  • Osteoblasts / drug effects
  • Osteoblasts / metabolism*
  • Solutions
  • Thapsigargin / pharmacology

Substances

  • Calcium Channels
  • Enzyme Inhibitors
  • Indicators and Reagents
  • Ionophores
  • Solutions
  • Lead
  • Calcimycin
  • Thapsigargin
  • Calcium