Inhibition of c-Jun N-terminal kinase pathway attenuates cerebral vasospasm after experimental subarachnoid hemorrhage through the suppression of apoptosis

Acta Neurochir Suppl. 2008:104:27-31. doi: 10.1007/978-3-211-75718-5_6.

Abstract

Background: Recent studies have demonstrated that apoptosis in cerebral arteries could play an essential role in cerebral vasospasm after subarachnoid hemorrhage (SAH) and that SP600125, an inhibitor of c-Jun N-terminal kinase (JNK) could suppress apoptosis. The present study examined whether SP600125 could reduce cerebral vasospasm through the suppression of apoptosis.

Method: Fifteen dogs were assigned to 3 groups: control, SAH, and SAH + SP600125 (30 micromol/l). SAH was induced by the injection of autologous blood into the cisterna magna on day 0 and day 2. Angiograms were evaluated on day 0 and day 7. The activation of the JNK pathway and caspase-3 were also evaluated using Western blot. To determine the distribution, TUNEL staining and immunohistochemistry for phosphorylated c-jun and cleaved caspase-3 were performed.

Findings: Severe vasospasm was observed in the basilar artery of the SAH dogs. SP600125 reduced angiographic and morphological vasospasm and reduced the expression of cleaved caspase-3, thereby suppressing apoptosis.

Conclusions: These results demonstrate that SP600125 attenuates cerebral vasospasm through the suppression of apoptosis, which may provide a novel therapeutic target for cerebral vasospasm.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anthracenes / therapeutic use*
  • Apoptosis / drug effects*
  • Basilar Artery / drug effects
  • Basilar Artery / pathology
  • Basilar Artery / physiopathology
  • Disease Models, Animal
  • Dogs
  • JNK Mitogen-Activated Protein Kinases / antagonists & inhibitors*
  • Subarachnoid Hemorrhage / pathology*
  • Vasospasm, Intracranial / pathology
  • Vasospasm, Intracranial / physiopathology*

Substances

  • Anthracenes
  • pyrazolanthrone
  • JNK Mitogen-Activated Protein Kinases