A soluble activin type IIA receptor induces bone formation and improves skeletal integrity

Proc Natl Acad Sci U S A. 2008 May 13;105(19):7082-7. doi: 10.1073/pnas.0711263105. Epub 2008 May 6.

Abstract

Diseases that affect the regulation of bone turnover can lead to skeletal fragility and increased fracture risk. Members of the TGF-beta superfamily have been shown to be involved in the regulation of bone mass. Activin A, a TGF-beta signaling ligand, is present at high levels in bone and may play a role in the regulation of bone metabolism. Here we demonstrate that pharmacological blockade of ligand signaling through the high affinity receptor for activin, type II activin receptor (ActRIIA), by administration of the soluble extracellular domain of ActRIIA fused to a murine IgG2a-Fc, increases bone formation, bone mass, and bone strength in normal mice and in ovariectomized mice with established bone loss. These observations support the development of this pharmacological strategy for the treatment of diseases with skeletal fragility.

MeSH terms

  • Activin Receptors, Type II / administration & dosage
  • Activin Receptors, Type II / isolation & purification
  • Activin Receptors, Type II / pharmacology*
  • Animals
  • Biomechanical Phenomena
  • Bone Resorption
  • Bone and Bones / drug effects*
  • Cell Line
  • Female
  • Humans
  • Immunoglobulin G / administration & dosage
  • Immunoglobulin G / isolation & purification
  • Immunoglobulin G / pharmacology
  • Lumbar Vertebrae / drug effects
  • Mice
  • Organ Size / drug effects
  • Osteogenesis / drug effects*
  • Ovariectomy
  • Recombinant Fusion Proteins / administration & dosage
  • Recombinant Fusion Proteins / isolation & purification
  • Recombinant Fusion Proteins / pharmacology
  • Solubility / drug effects

Substances

  • Immunoglobulin G
  • Recombinant Fusion Proteins
  • Activin Receptors, Type II
  • activin receptor type II-A