IL-8 as antibody therapeutic target in inflammatory diseases: reduction of clinical activity in palmoplantar pustulosis

J Immunol. 2008 Jul 1;181(1):669-79. doi: 10.4049/jimmunol.181.1.669.

Abstract

IL-8 is a chemokine that has been implicated in a number of inflammatory diseases involving neutrophil activation. HuMab 10F8 is a novel fully human mAb against IL-8, which binds a discontinuous epitope on IL-8 overlapping the receptor binding site, and which effectively neutralizes IL-8-dependent human neutrophil activation and migration. We investigated whether interference in the cytokine network by HuMab 10F8 might benefit patients suffering from palmoplantar pustulosis, a chronic inflammatory skin disease. Treatment of patients with HuMab 10F8 was well tolerated and significantly reduced clinical disease activity at all five endpoints, which included a >or=50% reduction in the formation of fresh pustules. IL-8 neutralization was monitored at the site of inflammation by assessing exudates of palmoplantar pustulosis lesions. HuMab 10F8 sequestered IL-8 in situ, as observed by rapid dose-dependent decreases of IL-8 concentrations immediately following Ab infusion. These data demonstrate a critical role for IL-8 in the pathophysiology of palmoplantar pustulosis. HuMab 10F8 is capable of interrupting IL-8 activity in vivo and represents a candidate for treatment of inflammatory diseases and other pathological conditions associated with IL-8 overproduction.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antibodies, Monoclonal / adverse effects
  • Antibodies, Monoclonal / blood
  • Antibodies, Monoclonal / immunology*
  • Antibodies, Monoclonal / therapeutic use*
  • Cells, Cultured
  • Epitopes / chemistry
  • Epitopes / immunology
  • Humans
  • Immune Tolerance / immunology
  • Immunotherapy
  • Inflammation / drug therapy
  • Inflammation / immunology
  • Inflammation / pathology
  • Interleukin-8 / chemistry
  • Interleukin-8 / immunology*
  • Mice
  • Mice, Transgenic
  • Models, Molecular
  • Molecular Sequence Data
  • Neutrophils / immunology
  • Protein Binding
  • Protein Structure, Tertiary
  • Psoriasis / drug therapy*
  • Psoriasis / immunology*
  • Psoriasis / pathology
  • Time Factors

Substances

  • Antibodies, Monoclonal
  • Epitopes
  • Interleukin-8