[Effects of valsartan on the renal vascular endothelial growth factor and its receptor flk-1 of diabetic rats]

Sichuan Da Xue Xue Bao Yi Xue Ban. 2008 Mar;39(2):223-6, 230.
[Article in Chinese]

Abstract

Objective: To explore effects of valsartan on expression changes of vascular endothelial growth factor (VEGF) and its receptor Flk-1 in diabetic rat kidney.

Methods: To establish the diabetic nephropathy (DN) rat models and divide the experiment rats into three groups--the DN group, the valsartan group and the control group, and use the reverse transcriptase polymerase chain reaction (RT-PCR), Western Blotting and immunohistochemical techniques to detect the expression of VEGF and Flk-1, and detect the urine protein and glomerular area and volume, then analyze the relationship of the data.

Results: The mRNA and protein expression of VEGF and Flk-1, the urine protein and glomerular area and volume in the DN were higher than those in the control group and valsartan group (P < 0.05). VEGF and Flk-1 were positively correlated with the urine protein and glomerular area and volume (P < 0.05).

Conclusion: VEGF and Flk-1 play an important role in the pathogenesis of DN, of which over-expression may lead to the damage of kidney. The angiotensin II receptor antagonist--valsartan can protect kidney through the non-hemodynamic mechanism of inhibiting the abnormal expression of VEGF and Flk-1.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Antihypertensive Agents / pharmacology
  • Blotting, Western
  • Diabetes Mellitus, Experimental / physiopathology*
  • Immunohistochemistry
  • Kidney / drug effects*
  • Kidney / metabolism
  • Kidney / pathology
  • Male
  • RNA, Messenger / biosynthesis
  • RNA, Messenger / genetics
  • Rats
  • Rats, Sprague-Dawley
  • Reverse Transcriptase Polymerase Chain Reaction
  • Tetrazoles / pharmacology*
  • Valine / analogs & derivatives*
  • Valine / pharmacology
  • Valsartan
  • Vascular Endothelial Growth Factor A / biosynthesis*
  • Vascular Endothelial Growth Factor A / genetics
  • Vascular Endothelial Growth Factor Receptor-1 / biosynthesis*
  • Vascular Endothelial Growth Factor Receptor-1 / genetics

Substances

  • Antihypertensive Agents
  • RNA, Messenger
  • Tetrazoles
  • Vascular Endothelial Growth Factor A
  • Valsartan
  • Flt1 protein, rat
  • Vascular Endothelial Growth Factor Receptor-1
  • Valine