Direct inhibitory effect of amino-terminal parathyroid hormone fragment [PTH(1-34)] on PTH secretion from bovine parathyroid primary cultured cells in vitro

Biochem Biophys Res Commun. 1991 Aug 15;178(3):953-8. doi: 10.1016/0006-291x(91)90984-f.

Abstract

We have examined the possibility of direct inhibitory effect of PTH(1-34) on PTH secretion in bovine parathyroid cells. As low as 10(-12) M PTH(1-34) completely inhibited low calcium (0.5 mM Ca2+)-stimulated PTH secretion by these cells. In the presence of 1.25 mM Ca2+, 10(-12) M PTH(1-34) inhibited PTH secretion by about 14.3% of the basal value, while 10(-11) M or higher concentration of PTH(1-34) showed potent inhibitory effects equivalent to the inhibitory action of high calcium concentration (2.5 mM Ca2+) on PTH secretion. At 2.5 mM Ca2+, as much as 10(-9) M PTH(1-34) failed to inhibit PTH secretion further. These results suggest that PTH(1-34) might directly, not via calcium concentration, inhibit PTH secretion by parathyroid cells and that a cooperative mechanism could exist between calcium and PTH(1-34) to inhibit PTH secretion.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium / pharmacology
  • Cattle
  • Cells, Cultured
  • Dose-Response Relationship, Drug
  • Kinetics
  • Parathyroid Glands / drug effects
  • Parathyroid Glands / metabolism*
  • Parathyroid Hormone / antagonists & inhibitors
  • Parathyroid Hormone / metabolism*
  • Parathyroid Hormone / pharmacology*
  • Peptide Fragments / pharmacology*
  • Teriparatide
  • Time Factors

Substances

  • Parathyroid Hormone
  • Peptide Fragments
  • Teriparatide
  • Calcium