Stereoselective synthesis of L-guluronic acid alginates

Chemistry. 2008;14(30):9400-11. doi: 10.1002/chem.200800960.

Abstract

The glycosylation properties of gulopyranosides have been mapped out, and it is shown that gulose has an intrinsic preference for the formation of 1,2-cis-glycosidic bonds. It is postulated that this glycosylation behaviour originates from nucleophilic attack at the oxacarbenium ion, which adopts the most favourable 3H4 conformation. Building on the stereoselectivity of gulose, a guluronic acid alginate trisaccharide was assembled for the first time by using gulopyranosyl building blocks.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alginates / chemical synthesis*
  • Alginates / chemistry
  • Esters / chemistry
  • Glucose / chemistry
  • Glycosylation
  • Hexuronic Acids / chemistry*
  • Stereoisomerism
  • Substrate Specificity

Substances

  • Alginates
  • Esters
  • Hexuronic Acids
  • guluronic acid
  • Glucose