The IKK-neutralizing compound Bay11 kills supereffector CD8 T cells by altering caspase-dependent activation-induced cell death

J Leukoc Biol. 2009 Jan;85(1):175-85. doi: 10.1189/jlb.0408248. Epub 2008 Oct 15.

Abstract

Antigen with dual costimulation through CD137 and CD134 induces powerful CD8 T cell responses. These effector T cells are endowed with an intrinsic survival program resulting in their accumulation in vivo, but the signaling components required for survival are unknown. We tested a cadre of pathway inhibitors and found one preclinical compound, Bay11-7082 (Bay11), which prevented survival. Even the gammac cytokine family members IL-2, -4, -7, and -15 could not block death, nor could pretreatment with IL-7. We found that dual costimulation caused loading of phosphorylated IkappaBalpha (p-IkappaBalpha) and high basal levels of NF-kappaB activity in the effector CD8 T cells. Bay11 trumped both events by reducing the presence of p-IkappaBalpha and ensuing NF-kappaB activity. Not all pathways were impacted to this degree, however, as mitogen-mediated ERK phosphorylation was evident during NF-kappaB inhibition. Nonetheless, Bay11 blocked TCR-stimulated cytokine synthesis by rapidly accentuating activation-induced cell death through elicitation of a caspase-independent pathway. Thus, in effector CD8 T cells, Bay11 forces a dominant caspase-independent death signal that cannot be overcome by an intrinsic survival program nor by survival-inducing cytokines. Therefore, Bay11 may be a useful tool to deliberately kill death-resistant effector T cells for therapeutic benefit.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • CD8-Positive T-Lymphocytes / drug effects
  • CD8-Positive T-Lymphocytes / immunology
  • CD8-Positive T-Lymphocytes / physiology*
  • Caspase 3 / metabolism*
  • Caspase 8 / metabolism*
  • Cell Survival
  • Cells, Cultured
  • Cytokines / biosynthesis
  • Enzyme Activation
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • I-kappa B Kinase / antagonists & inhibitors
  • I-kappa B Kinase / metabolism*
  • Mice
  • Mice, Inbred C57BL
  • NF-kappa B / antagonists & inhibitors
  • NF-kappa B / metabolism
  • Nitriles / pharmacology*
  • Peptides / pharmacology
  • Phosphorylation
  • Receptors, OX40 / metabolism
  • Sulfones / pharmacology*
  • Tumor Necrosis Factor Receptor Superfamily, Member 9 / immunology

Substances

  • 3-(4-methylphenylsulfonyl)-2-propenenitrile
  • Cytokines
  • NF-kappa B
  • Nitriles
  • Peptides
  • Receptors, OX40
  • Sulfones
  • Tnfrsf4 protein, mouse
  • Tumor Necrosis Factor Receptor Superfamily, Member 9
  • I-kappa B Kinase
  • Extracellular Signal-Regulated MAP Kinases
  • Casp8 protein, mouse
  • Caspase 3
  • Caspase 8