HSP27 regulates IL-1 stimulated IKK activation through interacting with TRAF6 and affecting its ubiquitination

Cell Signal. 2009 Jan;21(1):143-50. doi: 10.1016/j.cellsig.2008.10.001. Epub 2008 Oct 10.

Abstract

Heat shock protein 27 (HSP27) is an ubiquitiously expressed protein, which has been mediated in various biological functions. Here, we present a novel mechanism utilized by HSP27 in regulating IL-1beta induced NF-small ka, CyrillicB activation. Both over-expression and RNAi experiments indicate that HSP27 physically interacts with tumor necrosis factor receptor-associated factor 6 (TRAF6) and promotes TRAF6 ubiquitination. Over-expressed HSP27 augments IL-1beta induced TRAF6 ubiquitination and Ismall ka, CyrillicB kinase (IKK) activation. On the other hand, IL-1beta stimulation reduces endogenous HSP27/TRAF6 association, but inhibiting HSP27 phosphorylation by using SB202190, an inhibitor of p38, and MAPKAPK2 RNAi increases HSP27/TRAF6 association and thereby enhances TRAF6 ubiquitination, IKK phosphorylation as well as NF-small ka, CyrillicB activation. Furthermore, co-transfection study shows that HSP27 S78/82A, two phosphorylated serine site deficient mutants, but not wild-type HSP27 (HSP27 WT) and HSP27 S15A mutant increases TRAF6 ubiquitination and thereby mediates IL-1beta triggered IKK phosphorylation. Taken together, our data indicate that HSP27 regulates IL-1beta triggered NF-small ka, CyrillicB activation via a feedback loop which includes the interaction between HSP27 phosphorylation and ability of HSP27 to bind with TRAF6. The findings of this study reveal a novel mechanism by which HSP27 controls cytokine stimulation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line
  • HSP27 Heat-Shock Proteins / genetics
  • HSP27 Heat-Shock Proteins / metabolism*
  • I-kappa B Kinase / metabolism*
  • Immunoprecipitation
  • Interleukin-1beta / metabolism*
  • Intracellular Signaling Peptides and Proteins / metabolism
  • Mutagenesis, Site-Directed
  • NF-kappa B / metabolism
  • Phosphorylation
  • Protein Serine-Threonine Kinases / metabolism
  • RNA, Small Interfering / genetics
  • Signal Transduction
  • TNF Receptor-Associated Factor 6 / metabolism*
  • Ubiquitination*
  • p38 Mitogen-Activated Protein Kinases / metabolism

Substances

  • HSP27 Heat-Shock Proteins
  • Interleukin-1beta
  • Intracellular Signaling Peptides and Proteins
  • NF-kappa B
  • RNA, Small Interfering
  • TNF Receptor-Associated Factor 6
  • MAP-kinase-activated kinase 2
  • Protein Serine-Threonine Kinases
  • I-kappa B Kinase
  • p38 Mitogen-Activated Protein Kinases