Synthesis and anti-inflammatory and analgesic activities of phenoxyalkanoic acid derivatives

Arch Pharm Res. 1997 Feb;20(1):72-5. doi: 10.1007/BF02974045.

Abstract

The synthesis of phenoxyalkanoic acid derivatives and their anti-inflammatory and analgesic activities are described. Analysis of structure-activity relationships shows that in trichlorophenoxy derivatives anti-edematous potency is associated with the presence of 1-thiopropyl moiety and 2 or 4-aminopyridyl moiety at R' position contributes to the analgesic activity.