Kinetic analysis of salting activation of a subtilisin-like halophilic protease

Biochim Biophys Acta. 2009 Feb;1794(2):367-73. doi: 10.1016/j.bbapap.2008.10.017. Epub 2008 Nov 12.

Abstract

The secreted extracellular subtilase SR5-3 from Halobacillus sp. bacterium, isolated from the high-salt environment of Thai fish sauce, was utilized as a model halophilic serine protease. The dependence of salt activation on the size and structure of substrates was evaluated assaying the enzyme with Suc-AAPF-MCA and with the Fluorescence Resonance Energy Transfer (FRET) peptide Abz-AAPFSSKQ-EDDnp. Solvent isotope effects (SIE) and the thermodynamic parameters for activation of the hydrolysis of Suc-AAPF-MCA and Abz-AAPFSSKQ-EDDnp by SR5-3 protease in the presence of salts were also performed. All the obtained results support the notion that the salting out effect is responsible for the halophilic character of SR5-3, and the magnitude of its hydrolytic activity is mainly derived from the improvement of catalytic and/or interaction steps depending on the nature and size of the substrates, principally if they occupy the substrate prime subsites.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Bacillaceae / enzymology*
  • Bacterial Proteins / chemistry
  • Bacterial Proteins / metabolism*
  • Catalysis
  • Enzyme Activation
  • Fluorescence Resonance Energy Transfer
  • Hydrogen-Ion Concentration
  • Hydrolysis
  • Kinetics
  • Salts / chemistry
  • Salts / pharmacology*
  • Serine Endopeptidases / chemistry
  • Serine Endopeptidases / metabolism*
  • Subtilisin / chemistry
  • Subtilisin / metabolism*
  • Temperature

Substances

  • Bacterial Proteins
  • Salts
  • Serine Endopeptidases
  • Subtilisin