Olefin metathesis based approach to diversely functionalized pyrrolizidines and indolizidines; total synthesis of (+)-monomorine

J Org Chem. 2009 Jan 16;74(2):590-6. doi: 10.1021/jo801638u.

Abstract

New scaffolds for the stereoselective synthesis of diversely functionalized chiral enantiopure indolizidines and pyrrolizidines were synthesized from the cross and ring-closing metathesis reactions of appropriate intermediates, readily available from L-pyroglutamic acid. The versatility of this strategy was demonstrated by the synthesis of an indolizidine-based azasugar analogue and of the natural alkaloid (+)-monomorine.

MeSH terms

  • Alkenes / chemistry*
  • Indolizidines / chemical synthesis*
  • Indolizines / chemical synthesis*
  • Pyrrolizidine Alkaloids / chemical synthesis*
  • Stereoisomerism

Substances

  • Alkenes
  • Indolizidines
  • Indolizines
  • Pyrrolizidine Alkaloids
  • monomorine