15-HETE suppresses K(+) channel activity and inhibits apoptosis in pulmonary artery smooth muscle cells

Apoptosis. 2009 Jan;14(1):42-51. doi: 10.1007/s10495-008-0286-6.

Abstract

15-Hydroxyeicosatetraenoic acid (15-HETE) is an important hypoxic product from arachidonic acid (AA) in the wall of pulmonary vessels. Although its effects on pulmonary artery constriction are well known, it remains unclear whether 15-HETE acts on the apoptotic responses in pulmonary artery smooth muscle cells (PASMCs) and whether K(+) channels participate in this process. These hypothesises were validated by cell viability assay, terminal deoxynucleotidyl transferase-mediated dUTP nick end-labeling, mitochondrial potentials assay, caspase activity assay and western blot. We found that 15-HETE enhanced cell survival, suppressed the expression and activity of caspase-3, upregulated bcl-2 and attenuated mitochondrial depolarization, prevented chromatin condensation and partly reversed K(+) channel opener-induced apoptosis in PASMCs under serum-deprived conditions. Our data indicated that 15-HETE inhibits the apoptosis in PASMCs through, at least in part, inactivating K(+) channels.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis*
  • Arachidonic Acid / chemistry
  • Caspase 3 / metabolism
  • Humans
  • Hydrogen Peroxide / chemistry
  • Hydroxyeicosatetraenoic Acids / pharmacology*
  • Hypoxia
  • Mitochondria / metabolism
  • Models, Biological
  • Myocytes, Smooth Muscle / metabolism*
  • Potassium / chemistry
  • Potassium Channels / chemistry*
  • Proto-Oncogene Proteins c-bcl-2 / metabolism
  • Pulmonary Artery / pathology*
  • Tetrazolium Salts / pharmacology
  • Thiazoles / pharmacology

Substances

  • Hydroxyeicosatetraenoic Acids
  • Potassium Channels
  • Proto-Oncogene Proteins c-bcl-2
  • Tetrazolium Salts
  • Thiazoles
  • Arachidonic Acid
  • 15-hydroxy-5,8,11,13-eicosatetraenoic acid
  • Hydrogen Peroxide
  • Caspase 3
  • thiazolyl blue
  • Potassium