Construction of a functional lactose permease devoid of cysteine residues

Biochemistry. 1991 Oct 8;30(40):9595-600. doi: 10.1021/bi00104a005.

Abstract

By use of oligonucleotide-directed, site-specific mutagenesis, a lactose (lac) permease molecule was constructed in which all eight cysteinyl residues were simultaneously mutagenized (C-less permease). Cys154 was replaced with valine, and Cys117, -148, -176, -234, -333, -353, and -355 were replaced with serine. Remarkably, C-less permease catalyzes lactose accumulation in the presence of a transmembrane proton electrochemical gradient (interior negative and alkaline). Thus, in intact cells and right-side-out membrane vesicles containing comparable amounts of wild-type and Cys-less permease, the mutant protein catalyzes lactose transport at a maximum velocity and to a steady-state level of accumulation of about 35% and 55%, respectively, of wild-type with a similar apparent Km (ca. 0.3 mM). As anticipated, moreover, active lactose transport via C-less permease is completely resistant to inactivation by N-ethylmaleimide. Finally, C-less permease also catalyzes efflux and equilibrium exchange at about 35% of wild-type activity. The results provide definitive evidence that sulfhydryl groups do not play an essential role in the mechanism of lactose/H+ symport. Potential applications of the C-less mutant to studies of static and dynamic aspects of permease structure/function are discussed.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Base Sequence
  • Biological Transport
  • Cell Membrane / metabolism
  • Cysteine / genetics*
  • Escherichia coli / cytology
  • Escherichia coli / enzymology
  • Escherichia coli / genetics
  • Escherichia coli Proteins*
  • Genes, Bacterial
  • Lactose / metabolism
  • Membrane Transport Proteins / chemistry
  • Membrane Transport Proteins / genetics*
  • Molecular Sequence Data
  • Monosaccharide Transport Proteins*
  • Mutagenesis, Site-Directed*
  • Protein Conformation
  • Structure-Activity Relationship
  • Symporters*

Substances

  • Escherichia coli Proteins
  • LacY protein, E coli
  • Membrane Transport Proteins
  • Monosaccharide Transport Proteins
  • Symporters
  • lactose permease
  • Lactose
  • Cysteine