Prostatic soy isoflavone concentrations exceed serum levels after dietary supplementation

Prostate. 2009 May 15;69(7):719-26. doi: 10.1002/pros.20922.

Abstract

Background: The effects of soy isoflavones on prostate cancer may be concentration-dependent. The impact of soy supplementation on isoflavone concentrations in prostate tissues and serum remain unclear.

Objective: To assess and compare concentrations of soy isoflavones in prostate tissue and serum among 19 men with prostate cancer who had elected to undergo radical prostatectomy.

Methods: Participants were randomized to receive either daily soy supplements (82 mg/day aglycone equivalents) or placebos for 2 weeks (14 days) prior to surgery. Serum samples were obtained at the time of the surgery. Isoflavone concentrations were measured by HPLC/ESI-MS-MS.

Results: The median (25th, 75th percentile) total isoflavone concentration in the isoflavone-supplemented group was 2.3 micromol/L (1.2, 6.9) in the prostate tissue and 0.7 micromol/L (0.2, 1.2) in the serum. Total isoflavone concentrations in this group were an average of approximately 6-fold higher in prostate tissue compared to serum; the tissue versus serum ratio was significantly lower for genistein than daidzein, 4-fold versus 10-fold, P = 0.003. Tissue and serum levels of isoflavones among the placebo group were negligible with a few exceptions.

Conclusions: The findings from the present study suggest that prostate tissue may have the ability to concentrate dietary soy isoflavones to potentially anti-carcinogenic levels.

Publication types

  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, N.I.H., Extramural

MeSH terms

  • Adenocarcinoma / blood
  • Adenocarcinoma / metabolism*
  • Adenocarcinoma / surgery
  • Dietary Supplements
  • Double-Blind Method
  • Equol
  • Genistein / administration & dosage
  • Genistein / pharmacokinetics
  • Glycine max
  • Humans
  • Isoflavones / administration & dosage*
  • Isoflavones / blood
  • Isoflavones / pharmacokinetics*
  • Male
  • Mass Spectrometry
  • Prostatic Neoplasms / blood
  • Prostatic Neoplasms / metabolism*
  • Prostatic Neoplasms / surgery
  • Statistics, Nonparametric

Substances

  • 4',7-dihydroxy-3,4-dihydroisoflavone
  • Isoflavones
  • Equol
  • daidzein
  • Genistein