Current status of newer carbapenems

Curr Med Chem. 2009;16(5):564-75. doi: 10.2174/092986709787458498.

Abstract

Objectives: Beta-lactam antibiotics represent the most commonly prescribed antibacterial agents. Since many bacteria have developed resistance to older agents, new beta-lactams have been introduced constantly. In the late 1970s, a new class of exceptionally broad-spectrum beta-lactams, the carbapenems, was identified. The carbapenems, such as the most popular imipenem and meropenem, have the widest spectra of antibacterial activity of all the beta-lactams and provide excellent coverage of many gram-negative and gram-positive aerobic and anaerobic bacteria. Despite the wide antibacterial spectrum, the carbapenems globally lack activity against Enterococcus faecium, methicillin-resistant Staphylococcus aureus (MRSA) and Stenotrophomonas maltophilia.

Methods: We reviewed the principal characteristics of the novel carbapenems and their clinical implications.

Results and conclusions: We included in our review: ertapenem, biapenem, panipenem, doripenem, tebipenem pivoxil and tomopenem.

Publication types

  • Review

MeSH terms

  • Anti-Bacterial Agents / pharmacology*
  • Area Under Curve
  • Carbapenems / pharmacology*
  • Drug Resistance, Microbial

Substances

  • Anti-Bacterial Agents
  • Carbapenems