HIV-1 integrase polymorphisms are associated with prior antiretroviral drug exposure

Retrovirology. 2009 Feb 9:6:12. doi: 10.1186/1742-4690-6-12.

Abstract

In a recent summary of integrase sequences, primary integrase inhibitor mutations were rare. In a review of integrase inhibitor-naïve Australian HIV-1 sequences, primary mutations were not identified, although the accessory mutation G140S was detected. A link with previous antiretroviral therapy, intra-subtype B divergence across the integrase gene and transmission of integrase polymorphisms were also noted. Based on these findings, we would recommend ongoing surveillance of integrase mutations, and integrase region sequencing for patients prior to commencement of integrase inhibitors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-HIV Agents / therapeutic use*
  • Drug Resistance, Viral
  • HIV Infections / drug therapy*
  • HIV Infections / virology
  • HIV Integrase / genetics*
  • HIV Integrase / metabolism
  • HIV-1 / drug effects
  • HIV-1 / enzymology*
  • HIV-1 / genetics
  • Humans
  • Integrase Inhibitors / therapeutic use
  • Mutation
  • Polymorphism, Genetic*

Substances

  • Anti-HIV Agents
  • Integrase Inhibitors
  • HIV Integrase