D-serine, a selective glycine/N-methyl-D-aspartate receptor agonist, antagonizes the antidepressant-like effects of magnesium and zinc in mice

Pharmacol Rep. 2008 Nov-Dec;60(6):996-1000.

Abstract

Zinc and magnesium are potent inhibitors of the N-methyl-D-aspartate (NMDA) receptor complex. Recent data demonstrate that both zinc and magnesium, like other NMDA receptor antagonists, exhibit antidepressant-like activity in rodent screening tests and depression models. In the present study, we investigated the effect of D-serine (agonist for the glycine(B) site of the NMDA receptor complex; 100 nmol/mouse, icv) on magnesium (30 mg/kg, ip)- and zinc (5 mg/kg, ip)-induced activity during a forced swim test (FST) in mice. The antidepressant-like effect observed during FST for both ions was abolished by D-serine co-treatment. The present study indicates that the NMDA receptor complex, especially the glycine(B) site, plays a role in the antidepressant-like activity of magnesium and zinc in the FST in mice.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antidepressive Agents / pharmacology*
  • Magnesium / antagonists & inhibitors
  • Magnesium / pharmacology*
  • Male
  • Mice
  • Receptors, Glycine / agonists*
  • Receptors, Glycine / physiology
  • Receptors, N-Methyl-D-Aspartate / agonists*
  • Receptors, N-Methyl-D-Aspartate / physiology
  • Serine / pharmacology*
  • Zinc / antagonists & inhibitors
  • Zinc / pharmacology*

Substances

  • Antidepressive Agents
  • Receptors, Glycine
  • Receptors, N-Methyl-D-Aspartate
  • Serine
  • Magnesium
  • Zinc