Mdm2 affects genome stability independent of p53

Cancer Res. 2009 Mar 1;69(5):1697-701. doi: 10.1158/0008-5472.CAN-08-3732. Epub 2009 Feb 24.

Abstract

Mdm2 is a critical negative regulator of the p53 tumor suppressor and is frequently overexpressed in human cancers. However, reports, including our own studies, suggest that Mdm2 has both p53-dependent and p53-independent functions that contribute to genomic instability and transformation when deregulated. We recently elucidated a p53-independent role for Mdm2 in the regulation of the DNA double-strand break repair response, genomic stability, and transformation through interaction with Nbs1, a member of the Mre11/Rad50/Nbs1 DNA double-strand break repair complex. In light of these findings, targeting Mdm2 in human malignancies may have effects other than activating p53.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Cell Cycle Proteins / physiology
  • Cell Transformation, Neoplastic
  • DNA Breaks, Double-Stranded
  • DNA Repair
  • Genomic Instability*
  • Humans
  • Neoplasms / etiology*
  • Neoplasms / genetics
  • Nuclear Proteins / physiology
  • Proto-Oncogene Proteins c-mdm2 / physiology*
  • Tumor Suppressor Protein p53 / physiology*

Substances

  • Cell Cycle Proteins
  • NBN protein, human
  • Nuclear Proteins
  • Tumor Suppressor Protein p53
  • Proto-Oncogene Proteins c-mdm2