p53 acetylation is crucial for its transcription-independent proapoptotic functions

J Biol Chem. 2009 Apr 24;284(17):11171-83. doi: 10.1074/jbc.M809268200. Epub 2009 Mar 5.

Abstract

Acetylation of p53 at carboxyl-terminal lysine residues enhances its transcriptional activity associated with cell cycle arrest and apoptosis. Here we demonstrate that p53 acetylation at Lys-320/Lys-373/Lys-382 is also required for its transcription-independent functions in BAX activation, reactive oxygen species production, and apoptosis in response to the histone deacetylase inhibitors (HDACi) suberoylanilide hydroxamic acid and LAQ824. Knock-out of p53 markedly reduced HDACi-induced apoptosis. Unexpectedly, expression of transactivation-deficient p53 variants sensitized p53-null cells to HDACi-mediated BAX-dependent apoptosis, whereas knockdown of endogenous mutant p53 in cancer cells reduced HDACi-mediated cytotoxicity. Evaluation of the mechanisms controlling this response led to the discovery of a novel interaction between p53 and Ku70. The association between these two proteins was acetylation-independent, but acetylation of p53 could prevent and disrupt the Ku70-BAX complex and enhance apoptosis. These results suggest a new mechanism of acetylated p53 transcription-independent regulation of apoptosis.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antigens, Nuclear / biosynthesis
  • Apoptosis*
  • Cell Cycle
  • DNA-Binding Proteins / biosynthesis
  • Gene Expression Regulation, Neoplastic*
  • Glutathione Transferase / metabolism
  • Histone Deacetylases / metabolism
  • Humans
  • K562 Cells
  • Ku Autoantigen
  • Lysine / chemistry
  • Protein Structure, Tertiary
  • Subcellular Fractions
  • Transcription, Genetic*
  • Transcriptional Activation
  • Tumor Suppressor Protein p53 / metabolism*
  • bcl-2-Associated X Protein / metabolism

Substances

  • Antigens, Nuclear
  • DNA-Binding Proteins
  • TP53 protein, human
  • Tumor Suppressor Protein p53
  • bcl-2-Associated X Protein
  • Glutathione Transferase
  • Histone Deacetylases
  • Xrcc6 protein, human
  • Ku Autoantigen
  • Lysine