Downregulation of LRIG2 expression by RNA interference inhibits glioblastoma cell (GL15) growth, causes cell cycle redistribution, increases cell apoptosis and enhances cell adhesion and invasion in vitro

Cancer Biol Ther. 2009 Jun;8(11):1018-23. doi: 10.4161/cbt.8.11.8375. Epub 2009 Jun 10.

Abstract

The leucine-rich and immunoglobulin-like domains (LRIG) gene family contains LRIG1, 2 and 3. LRIG1 is a negative regulator of EGFR, but little is known about the function of LRIG2. To determine the role of LRIG2 in the progression of glioma, we performed RNA interference-mediated knockdown of LRIG2 in a human glioma cell line (GL15). Downregulation of LRIG2 expression resulted in: rapid EGF-mediated loss of EGFR; decreased proliferation; G(0)/G(1) arrest; increased spontaneous apoptosis; enhanced cell adhesion and increased invasion capability of GL15 cells in vitro. These findings indicate that LRIG2 possesses distinct functions compared with LRIG1 and validate the attractiveness of LRIG2 as a target in glioma therapy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis / genetics
  • Cell Adhesion / genetics
  • Cell Cycle / genetics
  • Cell Line, Tumor
  • Central Nervous System Neoplasms / genetics*
  • Central Nervous System Neoplasms / pathology
  • Down-Regulation
  • Epidermal Growth Factor / pharmacology
  • ErbB Receptors / biosynthesis
  • ErbB Receptors / genetics
  • Glioblastoma / genetics*
  • Glioblastoma / pathology
  • Humans
  • Membrane Glycoproteins / biosynthesis
  • Membrane Glycoproteins / deficiency
  • Membrane Glycoproteins / genetics*
  • RNA Interference
  • RNA, Neoplasm / genetics
  • RNA, Small Interfering / genetics*
  • Transfection

Substances

  • LRIG2 protein, human
  • Membrane Glycoproteins
  • RNA, Neoplasm
  • RNA, Small Interfering
  • Epidermal Growth Factor
  • ErbB Receptors