Comparative bioavailability of rectal and oral formulations of chloroquine

Pharm Weekbl Sci. 1991 Aug 23;13(4):176-8. doi: 10.1007/BF01957742.

Abstract

The relative bioavailability of chloroquinone in Witepsol H15 suppositories can vary between 10 and 53% of the bioavailability of a tablet formulation in adults. Therefore, it is therapeutically not sound to replace chloroquine tablets by a rectal formulation with the same dose.

Publication types

  • Comparative Study

MeSH terms

  • Administration, Oral
  • Administration, Rectal
  • Adult
  • Biological Availability
  • Chloroquine / administration & dosage
  • Chloroquine / pharmacokinetics*
  • Female
  • Humans
  • Male
  • Middle Aged

Substances

  • Chloroquine