Palladium-catalyzed direct arylation of cyclic enamides with aryl silanes by sp(2) C-H activation

Angew Chem Int Ed Engl. 2009;48(29):5355-7. doi: 10.1002/anie.200901884.

Abstract

It does get in! A fluoride-assisted direct cross-coupling of cyclic enamides with trialkoxy aryl silanes by a palladium-catalyzed C--H activation leads to a wide range of enamides in yields of up to 95 %.