Preventive effects of oligomerized polyphenol on estradiol-induced prostatitis in rats

Yonsei Med J. 2009 Jun 30;50(3):391-8. doi: 10.3349/ymj.2009.50.3.391. Epub 2009 Jun 23.

Abstract

Purpose: Chronic prostatitis/chronic pelvic pain syndrome (CP/CPPS, NIH category III) accounts for 90-95% of prostatitis cases. However, standard treatment has not yet been established. It is known that polyphenols have an inhibitory effect on inflammation by their antioxidative capacity, and oligonol, a polyphenol derivative, has much higher bioavailability and bioactivity than common polyphenols. We investigated the anti-inflammatory effects and mechanisms of oligonol in estradiol-induced prostatitis rat models.

Materials and methods: Prostatitis was induced by 17 beta-estradiol (E2) and dihydrotestosterone (DHT) in Wistar male rats (n = 20). Ten rats were placed in the oligonol-treated group and 10 in the E2 + DHT-treated group. The other 10 rats were also included as normal control group. Oligonol (60 mg/kg/day) was administered via gavage tube for 4 weeks. Superoxide dismutase (SOD), glutathione peroxidase (GPx), and tumor necrosis factor-alpha (TNF-alpha) were quantified, and phosphorylation of IkappaBa and histological changes were also evaluated in prostatic tissue.

Results: The SOD and GPx activity showed tendencies to increase in the oligonol-treated group compared to the normal control group. TNF-alpha expression was slightly reduced in the oligonol-treated group. Western blotting demonstrated that phosphorylation of IkappaBa in the oligonol-treated group was significantly lower than in the normal control group. The E2 + DHT-treated group revealed severe atrophy of acinar epithelial cells and infiltration of leukocytes and lymphocytes in the prostate, however, the oligonol-treated group showed overall reduction in inflammatory features.

Conclusion: This study demonstrates that oligonol improves estradiol-induced non-bacterial prostatitis by regulating phosphorylation of IkappaBa. These findings suggest that oligonol has a beneficial effect on prevention and treatment of CP/CPPS.

Keywords: Nonbacterial prostatitis; inflammation; oligonol; oxidative stress; polyphenol.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blotting, Western
  • Body Weight / drug effects
  • Estradiol / adverse effects*
  • Flavonoids / therapeutic use*
  • Immunoassay
  • Male
  • Phenols / therapeutic use*
  • Polyphenols
  • Prostate / drug effects
  • Prostate / pathology
  • Prostatitis / chemically induced*
  • Prostatitis / metabolism
  • Prostatitis / prevention & control*
  • Rats
  • Rats, Wistar
  • Superoxide Dismutase / metabolism
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Flavonoids
  • Phenols
  • Polyphenols
  • Tumor Necrosis Factor-alpha
  • Estradiol
  • Superoxide Dismutase