Application of a reservoir-type calcitriol transdermal patch in dairy cattle

J Vet Med Sci. 2009 Jun;71(6):845-8. doi: 10.1292/jvms.71.845.

Abstract

Our objective was to evaluate the effects of a reservoir-type calcitriol (5 mg/animal) transdermal patch on plasma calcitriol and calcium (Ca) concentrations in dairy cattle. A group of six heifers received three different types of patches: an encapsulated reservoir solution containing calcitriol alone (CAL), calcitriol with dodecylamine (CAL+D), or vehicle (CONT). The patches were applied to the skin of the tail for duration of 2 days at intervals of at least 3 weeks. Cattle that received CAL or CAL+D showed significant increases in plasma calcitriol and Ca concentrations on day 2 and days 2 and 3, respectively. The areas under the plasma concentration-time curve (AUC) values for plasma calcitriol and Ca in the CAL and CAL+D groups increased significantly compared to the CONT group. The data of this study describe evidence of measurable transdermal absorption of exogenous calcitriol from a patch and its sufficient biological action to elevate plasma Ca concentrations.

MeSH terms

  • Administration, Cutaneous
  • Amines / administration & dosage*
  • Amines / pharmacokinetics
  • Animals
  • Area Under Curve
  • Calcitriol / administration & dosage*
  • Calcitriol / blood
  • Calcitriol / pharmacokinetics
  • Calcium / blood
  • Cattle / blood
  • Cattle / metabolism*
  • Female
  • Random Allocation
  • Surface-Active Agents / administration & dosage*
  • Surface-Active Agents / pharmacokinetics
  • Vitamins / administration & dosage*
  • Vitamins / blood
  • Vitamins / pharmacokinetics

Substances

  • Amines
  • Surface-Active Agents
  • Vitamins
  • Calcitriol
  • Calcium
  • dodecylamine