A novel method for the encapsulation of biomolecules into polymersomes via direct hydration

Langmuir. 2009 Aug 18;25(16):9025-9. doi: 10.1021/la900779t.

Abstract

One of the major engineering challenges for the implementation of block copolymer vesicles, or polymersomes, as therapeutic drug carriers is obtaining high encapsulation efficiencies for biomolecules. Here we present a novel method for encapsulation of proteins with high encapsulation efficiency within polymersomes formed from block copolymers of poly(ethylene glycol)-bl-poly(propylene sulfide). By formulation of the neat block copolymer with a low molecular weight poly(ethylene glycol), direct hydration of the formulated mixture yielded polymersomes. We were able to achieve encapsulation efficiencies for ovalbumin at 37%, bovine serum albumin at 19%, and bovine gamma-globulin at 15% when the proteins were included in the hydration solution. The formulation process and the dispersion of polymersomes from the preparation in phosphate-buffered saline were characterized using confocal microscopy, cryogenic transmission electron microscopy, and fluorimetry. We were also successful in the encapsulation of proteinase K, a proteolytic enzyme, and demonstrated by SDS-PAGE that the enzyme was contained inside polymersomes when dispersed in a solution of ovalbumin.

MeSH terms

  • Animals
  • Capsules / chemistry*
  • Cattle
  • Microscopy, Confocal
  • Nanostructures / chemistry*
  • Polymers / chemistry*
  • Serum Albumin, Bovine / chemistry
  • Water / chemistry*

Substances

  • Capsules
  • Polymers
  • Water
  • Serum Albumin, Bovine