Distinct spatio-temporal Ca2+ signaling elicited by integrin alpha2beta1 and glycoprotein VI under flow

Blood. 2009 Sep 24;114(13):2793-801. doi: 10.1182/blood-2008-12-193490. Epub 2009 Jul 21.

Abstract

We studied how integrin alpha2beta1 and glycoprotein VI (GPVI) contribute to collagen-induced platelet activation under flow conditions by evaluating stable adhesion and intracellular Ca(2+) concentration ([Ca(2+)](i)) of FLUO 3-AM-labeled platelets perfused over acid-soluble type I or microfibrillar type VI collagen. Adhering platelets displayed 2 kinds of [Ca(2+)](i) oscillations. Rapid alpha-like peaks were unaffected by the membrane-impermeable Ca(2+) chelator ethyleneglycoltetraacetic acid but abolished by membrane-permeable BAPTA-AM. Longer-lasting gamma-like peaks were always preceded by at least one alpha-like peak and abolished by intracellular or extracellular Ca(2+) chelation. Inhibition of phosphatidylinositol 3-kinase or phospholipase C and modulation of cyclic nucleotides, but not blockage of adenosine diphosphate receptors, prevented both Ca(2+) responses. Human or mouse platelets lacking GPVI function exhibited alpha-like but not gamma-like Ca(2+) peaks, whereas those lacking alpha2beta1 showed markedly reduced to absent alpha-like and no gamma-like Ca(2+) peaks. Specific alpha2beta1 ligation induced alpha-like but not gamma-like peaks. Thus, alpha2beta1 may generate Ca(2+) signals that are reinforced by GPVI and required for subsequent longer-lasting Ca(2+) oscillation mediated by GPVI through transmembrane ion flux. Our results delineate a GPVI-independent signaling role of alpha2beta1 in response to collagen stimulation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blood Circulation / physiology*
  • Blood Platelets / drug effects
  • Blood Platelets / metabolism*
  • Blood Platelets / physiology
  • Calcium Signaling / drug effects
  • Calcium Signaling / genetics
  • Calcium Signaling / physiology*
  • Cells, Cultured
  • Chromones / pharmacology
  • Collagen Type I / metabolism
  • Collagen Type I / pharmacology
  • Enzyme Inhibitors / pharmacology
  • Humans
  • Integrin alpha2beta1 / genetics
  • Integrin alpha2beta1 / physiology*
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Morpholines / pharmacology
  • Phosphoinositide-3 Kinase Inhibitors
  • Platelet Adhesiveness / drug effects
  • Platelet Adhesiveness / genetics
  • Platelet Adhesiveness / physiology
  • Platelet Membrane Glycoproteins / genetics
  • Platelet Membrane Glycoproteins / physiology*
  • Time Factors

Substances

  • Chromones
  • Collagen Type I
  • Enzyme Inhibitors
  • Integrin alpha2beta1
  • Morpholines
  • Phosphoinositide-3 Kinase Inhibitors
  • Platelet Membrane Glycoproteins
  • platelet membrane glycoprotein VI
  • 2-(4-morpholinyl)-8-phenyl-4H-1-benzopyran-4-one