Increased efficacy of ganciclovir and foscarnet inhibition of cytomegalovirus replication in vitro by encapsulation in liposomes

Scand J Infect Dis Suppl. 1990:74:54-7.

Abstract

The antiviral effect of ganciclovir and foscarnet encapsulated in liposomes was studied against cytomegalovirus in human embryonic lung fibroblast cells. Substantially greater activity (3.5-fold and 38-fold respectively) in terms of inhibition of virus replication intracellularly was found compared to that seen with non-encapsulated antiviral agents, and liposome encapsulation did not result in increased cytotoxicity.

MeSH terms

  • Antiviral Agents / administration & dosage
  • Antiviral Agents / pharmacology*
  • Antiviral Agents / toxicity
  • Cells, Cultured
  • Cytomegalovirus / drug effects*
  • Cytomegalovirus / physiology
  • Drug Carriers
  • Fibroblasts / drug effects
  • Fibroblasts / microbiology
  • Foscarnet
  • Ganciclovir / administration & dosage
  • Ganciclovir / pharmacology*
  • Ganciclovir / toxicity
  • Humans
  • Liposomes
  • Phosphonoacetic Acid / administration & dosage
  • Phosphonoacetic Acid / analogs & derivatives*
  • Phosphonoacetic Acid / pharmacology
  • Phosphonoacetic Acid / toxicity
  • Viral Plaque Assay
  • Virus Replication / drug effects

Substances

  • Antiviral Agents
  • Drug Carriers
  • Liposomes
  • Foscarnet
  • Phosphonoacetic Acid
  • Ganciclovir