ROCK pathway participates in the processes that 15-hydroxyeicosatetraenoic acid (15-HETE) mediated the pulmonary vascular remodeling induced by hypoxia in rat

J Cell Physiol. 2010 Jan;222(1):82-94. doi: 10.1002/jcp.21923.

Abstract

15-Hydroxyeicosatetraenoic acid (15-HETE), a product of arachidonic acid (AA) catalyzed by 15-lipoxygenase (15-LO), plays an essential role in hypoxic pulmonary arterial hypertension. We have previously shown that 15-HETE inhibits apoptosis in pulmonary artery smooth muscle cells (PASMCs). To test the hypothesis that such an effect is attributable to the hypoxia-induced pulmonary vascular remodeling (PVR), we performed these studies. We found subtle thickening of proximal media/adventitia of the pulmonary arteries (PA) in rats that had been exposed to hypoxia. This was associated with an up-regulation of the anti-apoptotic Bcl-2 expression and down-regulation of pro-apoptotic caspase-3 and Bax expression in PA homogenates. Nordihydroguaiaretic acid (NDGA), which inhibits the generation of endogenous 15-HETE, reversed all the alterations following hypoxia. In situ hybridization histochemistry and immunocytochemistry showed that the 15-LO-1 mRNA and protein were localized in pulmonary artery endothelial cells (PAECs), while the 15-LO-2 mRNA and protein were localized in both PAECs and PASMCs. Furthermore, the Rho-kinase (ROCK) pathway was activated by both endogenous and exogenous 15-HETE, alleviating the serum deprivation (SD)-induced PASMC apoptosis. Thus, these findings indicate that 15-HETE protects PASMC from apoptosis, contributing to pulmonary vascular medial thickening, and the effect is, at least in part, mediated via the ROCK pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Arachidonate 15-Lipoxygenase / genetics
  • Arachidonate 15-Lipoxygenase / metabolism
  • Caspase 3 / metabolism
  • Cell Hypoxia / drug effects
  • Cell Survival / drug effects
  • DNA Fragmentation / drug effects
  • Down-Regulation / drug effects
  • Enzyme Activation / drug effects
  • Gene Expression Regulation, Enzymologic / drug effects
  • Hydroxyeicosatetraenoic Acids / pharmacology*
  • Isoenzymes / genetics
  • Isoenzymes / metabolism
  • Masoprocol / pharmacology
  • Membrane Potential, Mitochondrial / drug effects
  • Myocytes, Smooth Muscle / drug effects
  • Myocytes, Smooth Muscle / enzymology
  • Myocytes, Smooth Muscle / pathology
  • Organ Size / drug effects
  • Protein Kinase Inhibitors / pharmacology
  • Protein Transport / drug effects
  • Pulmonary Artery / drug effects
  • Pulmonary Artery / enzymology*
  • Pulmonary Artery / pathology*
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Rats
  • Signal Transduction / drug effects*
  • Subcellular Fractions / drug effects
  • Subcellular Fractions / enzymology
  • bcl-2-Associated X Protein / metabolism
  • rho-Associated Kinases / antagonists & inhibitors
  • rho-Associated Kinases / metabolism*

Substances

  • Hydroxyeicosatetraenoic Acids
  • Isoenzymes
  • Protein Kinase Inhibitors
  • RNA, Messenger
  • bcl-2-Associated X Protein
  • 15-hydroxy-5,8,11,13-eicosatetraenoic acid
  • Masoprocol
  • Arachidonate 15-Lipoxygenase
  • rho-Associated Kinases
  • Caspase 3