Doxorubicin-mediated apoptosis in glioma cells requires NFAT3

Cell Mol Life Sci. 2009 Dec;66(24):3967-78. doi: 10.1007/s00018-009-0157-5. Epub 2009 Sep 27.

Abstract

Nuclear factor of activated T cells (NFAT), a family of transcription factors, has been implicated in many cellular processes, including some cancers. Here, we characterize, for the first time, the role of NFAT3 in doxorubicin (DOX)-mediated apoptosis, migration, and invasion in SNB19 and U87 glioma cells. This study demonstrates that the specific knockdown of NFAT3 results in a dramatic inhibition of the apoptotic effect induced by DOX and favors cell survival. Inhibition of NFAT3 activation by shNFAT3 (shNF3) significantly downregulated tumor necrosis factor (TNF)-alpha induction, its receptor TNFR1, caspase 10, caspase 3, and poly (ADP-ribose) polymerase, abrogating DOX-mediated apoptosis in glioma cells. DOX treatment resulted in NFAT3 translocation to the nucleus. Similarly, shNF3 treatment in SNB19 and U87 cells reversed DOX-induced inhibition of cell migration and invasion, as determined by wound healing and matrigel invasion assays. Taken together, these results indicate that NFAT3 is a prerequisite for the induction of DOX-mediated apoptosis in glioma cells.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Active Transport, Cell Nucleus / drug effects
  • Antibiotics, Antineoplastic / pharmacology
  • Apoptosis / drug effects*
  • Blotting, Western
  • Caspase 10 / metabolism
  • Caspase 3 / metabolism
  • Cell Line, Tumor
  • Cell Movement / drug effects
  • Cell Nucleus / metabolism
  • Cell Survival / drug effects
  • Doxorubicin / pharmacology*
  • Flow Cytometry
  • Fluorescent Antibody Technique
  • G1 Phase / drug effects
  • Glioma / genetics
  • Glioma / metabolism
  • Glioma / pathology
  • Humans
  • NFATC Transcription Factors / genetics
  • NFATC Transcription Factors / metabolism
  • NFATC Transcription Factors / physiology*
  • Poly(ADP-ribose) Polymerases / metabolism
  • Protein Transport / drug effects
  • RNA Interference
  • Receptors, Tumor Necrosis Factor, Type I / metabolism
  • Resting Phase, Cell Cycle / drug effects
  • Reverse Transcriptase Polymerase Chain Reaction
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Antibiotics, Antineoplastic
  • NFATC Transcription Factors
  • Receptors, Tumor Necrosis Factor, Type I
  • Tumor Necrosis Factor-alpha
  • Doxorubicin
  • Poly(ADP-ribose) Polymerases
  • Caspase 10
  • Caspase 3