Synthetic peptides containing a conserved sequence motif of the Id protein family modulate vascular smooth muscle cell phenotype

Bioorg Med Chem Lett. 2009 Nov 15;19(22):6298-302. doi: 10.1016/j.bmcl.2009.09.105. Epub 2009 Oct 1.

Abstract

Modulation of smooth muscle cells to a proliferating and migrating phenotype with downregulated alpha-actin expression is observed upon vascular lesion formation. The Id proteins (inhibitors of cell differentiation) play a role in the development of this phenotype. In contrast, synthetic peptides based on a conserved 11-residue Id sequence trigger the switch to a contractile phenotype that shows reduced cell growth and migration, increased expression of alpha-actin and decreased Id protein levels.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actins / physiology
  • Amino Acid Motifs / physiology*
  • Aorta, Thoracic
  • Calcium-Binding Proteins
  • Cell Differentiation / physiology*
  • Cell Proliferation*
  • Conserved Sequence / physiology*
  • Endothelium, Vascular / cytology
  • Inhibitor of Differentiation Proteins / genetics
  • Inhibitor of Differentiation Proteins / physiology*
  • Muscle, Smooth, Vascular / physiology*
  • Myocytes, Smooth Muscle / cytology
  • Myocytes, Smooth Muscle / physiology
  • Nuclear Proteins
  • Peptides / chemical synthesis
  • Peptides / physiology*
  • Phenotype
  • Protein Binding
  • Repressor Proteins

Substances

  • Actins
  • Calcium-Binding Proteins
  • Inhibitor of Differentiation Proteins
  • Nuclear Proteins
  • Peptides
  • Repressor Proteins