A chemical platform for improved induction of human iPSCs

Nat Methods. 2009 Nov;6(11):805-8. doi: 10.1038/nmeth.1393. Epub 2009 Oct 18.

Abstract

The slow kinetics and low efficiency of reprogramming methods to generate human induced pluripotent stem cells (iPSCs) impose major limitations on their utility in biomedical applications. Here we describe a chemical approach that dramatically improves (200-fold) the efficiency of iPSC generation from human fibroblasts, within seven days of treatment. This will provide a basis for developing safer, more efficient, nonviral methods for reprogramming human somatic cells.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Benzamides / pharmacology
  • Cell Differentiation / genetics*
  • Dioxoles / pharmacology
  • Diphenylamine / analogs & derivatives
  • Diphenylamine / pharmacology
  • Fibroblasts / physiology
  • Humans
  • Induced Pluripotent Stem Cells / cytology*
  • Induced Pluripotent Stem Cells / physiology
  • MAP Kinase Kinase 1 / antagonists & inhibitors
  • Pyrimidines / pharmacology
  • Receptors, Transforming Growth Factor beta / antagonists & inhibitors
  • Thiazoles / pharmacology
  • Transduction, Genetic

Substances

  • 4-(5-benzo(1,3)dioxol-5-yl-4-pyridin-2-yl-1H-imidazol-2-yl)benzamide
  • Benzamides
  • Dioxoles
  • Pyrimidines
  • Receptors, Transforming Growth Factor beta
  • Thiazoles
  • thiazovivin
  • mirdametinib
  • Diphenylamine
  • MAP Kinase Kinase 1