Immune hemolytic anemia due to cimetidine: the first example of a cimetidine antibody

Transfusion. 2010 Feb;50(2):302-7. doi: 10.1111/j.1537-2995.2009.02447.x. Epub 2009 Oct 23.

Abstract

Background: Although there have been a few reports of immune hemolytic anemia (IHA) thought to be due to cimetidine, none of them provided proof (e.g., serologic detection of anti-cimetidine and/or repeat of IHA upon drug rechallenge). One report used cimetidine as an example of how temporal associations of drug administration and hemolytic anemia are not proof of a cause-effect relationship.

Study design and methods: A 63-year-old cancer patient developed IHA on two occasions after receiving cimetidine (with and without chemotherapy). Serologic methods included testing cimetidine-treated red blood cells (RBCs) as well as testing untreated RBCs in the presence of cimetidine.

Results: The patient's direct antiglobulin test was positive (C3 only) and a serum antibody to cimetidine was detected by both testing methods. An eluate from the patient's RBCs was nonreactive. Cimetidine-treated RBCs were optimally prepared at room temperature and needed to be tested on the day of preparation.

Conclusions: This is the first reported case of IHA due to a cimetidine antibody where a drug-dependent antibody was demonstrated. The patient had IHA after receiving cimetidine on two separate occasions.

Publication types

  • Case Reports

MeSH terms

  • Anemia, Hemolytic / chemically induced*
  • Anemia, Hemolytic / drug therapy
  • Anemia, Hemolytic / immunology
  • Anemia, Hemolytic / therapy
  • Antineoplastic Combined Chemotherapy Protocols / therapeutic use
  • Blood Transfusion
  • Breast Neoplasms / complications
  • Breast Neoplasms / drug therapy
  • Cimetidine / adverse effects*
  • Cimetidine / immunology
  • Combined Modality Therapy
  • Coombs Test
  • Dexamethasone / administration & dosage
  • Dexamethasone / therapeutic use
  • Diphenhydramine / administration & dosage
  • Diphenhydramine / therapeutic use
  • Erythrocyte Membrane / drug effects
  • Erythrocyte Membrane / immunology
  • Female
  • Histamine H2 Antagonists / administration & dosage
  • Histamine H2 Antagonists / immunology*
  • Histamine H2 Antagonists / therapeutic use
  • Humans
  • Immunoglobulin G / blood
  • Immunoglobulin G / immunology*
  • Immunoglobulin M / blood
  • Immunoglobulin M / immunology*
  • Immunosuppressive Agents / therapeutic use
  • Middle Aged
  • Models, Immunological
  • Prednisone / therapeutic use
  • Premedication

Substances

  • Histamine H2 Antagonists
  • Immunoglobulin G
  • Immunoglobulin M
  • Immunosuppressive Agents
  • Dexamethasone
  • Cimetidine
  • Diphenhydramine
  • Prednisone