Attenuation of adverse cardiac effects in prednisolone-treated delta-sarcoglycan-deficient mice by mineralocorticoid-receptor-antagonism

Neuromuscul Disord. 2010 Jan;20(1):21-8. doi: 10.1016/j.nmd.2009.10.003. Epub 2009 Nov 12.

Abstract

We have tested the hypothesis that the adverse effects of glucocorticoids in the delta-sarcoglycan-deficient (Sgcd-null) mouse are due to additional mineralocorticoid effects. We investigated the effects of spironolactone, an unselective mineralocorticoid-receptor antagonist, on in vivo cardiac haemodynamics, cardiomyocyte damage and fibrosis in prednisolone treated Sgcd-null mice. Oral spironolactone given to 8-week-old Sgcd-null non-steroid treated mice had beneficial effects on systolic function by improving myocardial contractility when assessed by pressure-volume loops. Given in combination with prednisolone, spironolactone prevented steroid-induced deterioration of cardiac haemodynamics and acute sarcolemmal damage but not cardiac fibrosis. This study demonstrates the beneficial effects of oral spironolactone on cardiac haemodynamics in Sgcd-null mice and its ability to prevent some of the adverse effects of glucocorticoids.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Animals
  • Body Weight / drug effects
  • Fibrosis / drug therapy
  • Glucocorticoids / adverse effects*
  • Glucocorticoids / therapeutic use
  • Heart / drug effects
  • Heart Diseases / chemically induced
  • Heart Diseases / drug therapy*
  • Heart Diseases / pathology
  • Hemodynamics / drug effects
  • Hormone Antagonists / administration & dosage
  • Hormone Antagonists / pharmacology*
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Mineralocorticoid Receptor Antagonists
  • Muscle Contraction / drug effects
  • Organ Size
  • Prednisolone / adverse effects*
  • Prednisolone / therapeutic use
  • Sarcoglycans / deficiency*
  • Sarcoglycans / genetics
  • Sarcolemma / drug effects
  • Spironolactone / administration & dosage
  • Spironolactone / pharmacology*

Substances

  • Glucocorticoids
  • Hormone Antagonists
  • Mineralocorticoid Receptor Antagonists
  • Sarcoglycans
  • Spironolactone
  • Prednisolone