[Calcium antagonists: current and future applications based on new evidence. Neuroprotective effect of calcium antagonists]

Clin Calcium. 2010 Jan;20(1):83-8.
[Article in Japanese]

Abstract

Voltage-dependent Ca(2+) channels have been divided into at least 5 types (L-, N-, T-, P-, and Q-type). L/N-type Ca(2+) channel blocker cilnidipine could reduce the size of cerebral infarction in the rat focal brain ischemia. L-type Ca(2+) channel blocker amlodipine reduced cerebral edema and inhibit neuronal cell death. N-type Ca(2+) channel blocker omega-conotoxin reduce the size of cerebral infarction and inhibit delayed neuronal cell death in hippocampal CA1 area. It is suggested that calcium antagonist has neuroprotective effect.

Publication types

  • English Abstract
  • Review

MeSH terms

  • Amlodipine / pharmacology*
  • Amlodipine / therapeutic use*
  • Animals
  • Brain Edema / drug therapy*
  • Calcium Channel Blockers / pharmacology*
  • Calcium Channel Blockers / therapeutic use*
  • Calcium Channels, L-Type
  • Calcium Channels, N-Type
  • Cell Death / drug effects
  • Cerebral Infarction / drug therapy*
  • Dihydropyridines / pharmacology*
  • Dihydropyridines / therapeutic use*
  • Hippocampus / cytology
  • Humans
  • Neurons / pathology
  • Neuroprotective Agents*
  • Rats
  • omega-Conotoxins / pharmacology*
  • omega-Conotoxins / therapeutic use*

Substances

  • Calcium Channel Blockers
  • Calcium Channels, L-Type
  • Calcium Channels, N-Type
  • Dihydropyridines
  • Neuroprotective Agents
  • omega-Conotoxins
  • Amlodipine
  • cilnidipine