Transcriptional activation of human MMP-13 gene expression by c-Maf in osteoarthritic chondrocyte

Connect Tissue Res. 2010;51(1):48-54. doi: 10.3109/03008200902989104.

Abstract

Matrix metalloproteinase (MMP)-13 has pivotal roles in the pathogenesis of Osteoarthritis (OA) and it is necessary to understand the regulatory mechanisms of MMP-13 expression. MMP-13 gene expression is regulated primarily at the transcriptional level. In this study, we investigated the role of c-maf in regulating MMP-13 transcription. Using transient transfection system with an c-maf construct, and MMP-13 promoter-luciferase constructs with specific mutations in transcription factor binding sites, we found that c-maf can significantly enhance MMP-13 promoter activity via the AP-1 site, By gene suppression with RNAi technology, we could show that c-maf downregulation leads to a reduced expression of MMP13. Chromatin immunoprecipitation assays reveal that c-maf binds to the MMP-13 gene promoter to a region of the MMP-13 promoter containing the AP-1 site. Taken together, these studies demonstrate a new level of transcriptional regulation of MMP-13 expression by the c-maf.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Binding Sites / genetics
  • Cartilage, Articular / metabolism*
  • Cartilage, Articular / pathology
  • Cartilage, Articular / physiopathology
  • Chondrocytes / cytology
  • Chondrocytes / metabolism*
  • DNA-Binding Proteins / genetics
  • Humans
  • Matrix Metalloproteinase 13 / genetics*
  • Osteoarthritis / genetics*
  • Osteoarthritis / metabolism*
  • Osteoarthritis / physiopathology
  • Promoter Regions, Genetic / genetics
  • Proto-Oncogene Proteins c-maf / genetics*
  • Transcription Factor AP-1 / genetics
  • Transcriptional Activation / genetics
  • Transfection

Substances

  • DNA-Binding Proteins
  • MAF protein, human
  • Proto-Oncogene Proteins c-maf
  • Transcription Factor AP-1
  • Matrix Metalloproteinase 13