Establishment and identification of the human multi-drug-resistant cholangiocarcinoma cell line QBC939/ADM

Mol Biol Rep. 2011 Jun;38(5):3075-82. doi: 10.1007/s11033-010-9975-7. Epub 2010 Jan 29.

Abstract

In this study, we aim to establish the human multi-drug-resistant cholangiocarcinoma cell line QBC939/ADM which can be grow and passaged steadily in 1 μg/ml concentration of adriamycin in appropriate medium. The human multi-drug-resistant cholangiocarcinoma cell line QBC939/ADM was established using the method of exposure to medium with adriamycin alternated between high and low concentration with gradually increasing concentration. Furthermore, QBC939 and QBC939/ADM were both treated with adriamycin, mitomycin and vindesine, and then detected by MTT assay, respectively. Growth cycle and intra-cellular concentrations of ADM within cells of each group were determined by flow cytometry. Expression levels of P-glycoprotein were detected by Western bolt and real-time PCR. Results showed that, compared with QBC939, the inhibitive rates of adriamycin, mitomycin and vindesine to QBC939/ADM were lower. Content of ADM in the QBC939/ADM was lower. Western bolt and real time PCR showed that P-glycoprotein in the QBC939/ADM group was over expressed. Therefore, QBC939/ADM was establish and identified as the multi-drug-resistant cell line, which can grow and be passaged steadily in 1 μg/ml concentration adriamycin in appropriate medium. And the multi-drug-resistant character of QBC939/ADM was indicated to be related to the over expression of P-glycoprotein induced by chemotherapeutic drugs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / metabolism
  • Antibiotics, Antineoplastic / pharmacology
  • Antineoplastic Agents, Phytogenic / pharmacology
  • Bile Duct Neoplasms / pathology*
  • Bile Duct Neoplasms / physiopathology*
  • Bile Ducts, Intrahepatic / pathology*
  • Cell Cycle / drug effects
  • Cell Line, Tumor / drug effects
  • Cell Line, Tumor / physiology*
  • Cholangiocarcinoma / pathology*
  • Cholangiocarcinoma / physiopathology*
  • Doxorubicin / pharmacology
  • Drug Resistance, Multiple / physiology*
  • Humans
  • Mitomycin / pharmacology
  • Vindesine / pharmacology

Substances

  • ATP Binding Cassette Transporter, Subfamily B, Member 1
  • Antibiotics, Antineoplastic
  • Antineoplastic Agents, Phytogenic
  • Mitomycin
  • Doxorubicin
  • Vindesine