Efficacy of moxidectin microsphere sustained release formulation for the prevention of subcutaneous filarial (Dirofilaria repens) infection in dogs

Vet Parasitol. 2010 May 28;170(1-2):167-9. doi: 10.1016/j.vetpar.2010.01.034. Epub 2010 Feb 2.

Abstract

A study was carried out to assess the efficacy of a moxidectin microsphere sustained release (SR) injectable formulation (Guardian SR Iniettabile, Fort Dodge) for the prevention of Dirofilaria repens infection in experimentally infected dogs. On day 0, 18 Beagle dogs, 9 male dogs and 9 female dogs, weighing 12-16 kg were ranked in ascending order of body weight (b.w.) and blocked into pairs. Within each pair, dogs were allocated to Group 1 or Group 2 at random. On the same day, dogs in Group 1 were injected with 0.05 ml/kg b.w. of saline solution and dogs in Group 2 were injected with moxidectin SR at the label dose 0.17 mg/kg b.w. (0.05 ml/kg b.w.). Six months after moxidectin SR or saline injection, on day 180, each dog in the two groups was challenged with 50 infective larvae of D. repens collected from laboratory-reared, experimentally infected Aedes aegypti. Dogs were humanely euthanized on day 380 of the study, approximately 7 months from D. repens challenge. At necropsy, no worms were found in dogs treated with moxidectin SR (Group 2) while adult worms were found in saline-treated dogs (total 90; 38 males and 52 females; arithmetic mean 10, standard error 0.96, median 9, range 7-15) (Group 1 vs Group 2 P<0.001). In this experimental study, moxidectin SR injectable showed full efficacy (100%) lasting at least 6 months, and is able to prevent subcutaneous D. repens patent infection throughout the entire transmission season in Europe.

MeSH terms

  • Animals
  • Anthelmintics / administration & dosage
  • Anthelmintics / pharmacology*
  • Anthelmintics / standards
  • Anthelmintics / therapeutic use
  • Delayed-Action Preparations / administration & dosage
  • Delayed-Action Preparations / pharmacology*
  • Delayed-Action Preparations / standards
  • Delayed-Action Preparations / therapeutic use
  • Dirofilaria / growth & development*
  • Dirofilariasis / drug therapy
  • Dirofilariasis / parasitology*
  • Dirofilariasis / prevention & control
  • Dog Diseases / drug therapy
  • Dog Diseases / parasitology*
  • Dog Diseases / prevention & control
  • Dogs
  • Female
  • Macrolides / administration & dosage
  • Macrolides / pharmacology
  • Macrolides / standards
  • Macrolides / therapeutic use
  • Male
  • Random Allocation
  • Statistics, Nonparametric

Substances

  • Anthelmintics
  • Delayed-Action Preparations
  • Macrolides
  • moxidectin