First characterization of the mutagenic specificity of 7-methoxy-2-nitronaphtho[2,1-b]furan (R7000) in Salmonella typhimurium

Mutat Res. 1991 May;248(1):85-92. doi: 10.1016/0027-5107(91)90090-b.

Abstract

In order to investigate the mutational events induced by the very potent genotoxic agent 7-methoxy-2-nitronaphtho[2,1-b]furan (R7000), we evaluated its mutagenic potency in a battery of his- mutants of Salmonella typhimurium designed to study mutagenic specificity (Levin and Ames, 1986). Using this system we could show that R7000 is able to induce base-pair substitutions, mainly GC----TA transversions and, perhaps to a lower extent, AT----TA transversions. In addition, our results suggest that this chemical may be a very efficient inducer of base-pair deletions/insertions resulting in frameshifts. Whereas the induction of base-pair substitutions by R7000 is dependent on the presence of plasmid pKM101 carrying the mucA,B operon, the induction of base-pair deletions/insertions is independent of the presence of the plasmid.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alanine / analogs & derivatives
  • Alanine / pharmacology
  • DNA Repair / drug effects
  • Drug Tolerance / genetics
  • Genes, Suppressor
  • Mutagenicity Tests
  • Mutagens*
  • Nitrofurans / pharmacology*
  • Salmonella typhimurium / drug effects
  • Salmonella typhimurium / genetics*

Substances

  • Mutagens
  • Nitrofurans
  • triazolealanine
  • 2-nitro-7-methoxynaphtho(2-1b)furan
  • Alanine