The effect of deuterium labeling on the genotoxicity of N-nitrosodimethylamine, epichlorohydrin and dimethyl sulfate

Mutat Res. 1991 May;263(1):9-12. doi: 10.1016/0165-7992(91)90027-2.

Abstract

Deuterated and non-deuterated N-nitrosodimethylamine, epichlorohydrin and dimethyl sulfate were evaluated for the ability to induce DNA single-strand breaks in rat hepatocytes as measured by alkaline elution. Non-deuterated nitrosodimethylamine induced twice the amount of DNA-strand breaks as the deuterated form. No evidence of a deuterium isotope effect was seen for the direct-acting alkylating agents epichlorohydrin and dimethyl sulfate.

MeSH terms

  • Animals
  • Cell Survival / drug effects
  • DNA Damage
  • Deuterium / chemistry*
  • Dimethylnitrosamine / toxicity*
  • Epichlorohydrin / toxicity*
  • Liver / cytology
  • Liver / drug effects*
  • Male
  • Mutagens*
  • Rats
  • Rats, Inbred Strains
  • Sulfuric Acid Esters / toxicity*

Substances

  • Mutagens
  • Sulfuric Acid Esters
  • Epichlorohydrin
  • Deuterium
  • dimethyl sulfate
  • Dimethylnitrosamine