Inflammation anergy in human intestinal macrophages is due to Smad-induced IkappaBalpha expression and NF-kappaB inactivation

J Biol Chem. 2010 Jun 18;285(25):19593-604. doi: 10.1074/jbc.M109.069955. Epub 2010 Apr 13.

Abstract

Human intestinal macrophages contribute to tissue homeostasis in noninflamed mucosa through profound down-regulation of pro-inflammatory cytokine release. Here, we show that this down-regulation extends to Toll-like receptor (TLR)-induced cytokine release, as intestinal macrophages expressed TLR3-TLR9 but did not release cytokines in response to TLR-specific ligands. Likely contributing to this unique functional profile, intestinal macrophages expressed markedly down-regulated adapter proteins MyD88 and Toll interleukin receptor 1 domain-containing adapter-inducing interferon beta, which together mediate all TLR MyD88-dependent and -independent NF-kappaB signaling, did not phosphorylate NF-kappaB p65 or Smad-induced IkappaBalpha, and did not translocate NF-kappaB into the nucleus. Importantly, transforming growth factor-beta released from intestinal extracellular matrix (stroma) induced identical down-regulation in the NF-kappaB signaling and function of blood monocytes, the exclusive source of intestinal macrophages. Our findings implicate stromal transforming growth factor-beta-induced dysregulation of NF-kappaB proteins and Smad signaling in the differentiation of pro-inflammatory blood monocytes into noninflammatory intestinal macrophages.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Cytokines / metabolism
  • Enzyme Inhibitors / chemistry
  • Gene Expression Regulation, Enzymologic*
  • Humans
  • I-kappa B Proteins / metabolism*
  • Inflammation*
  • Intestinal Mucosa / metabolism*
  • Macrophages / metabolism*
  • Monocytes / metabolism
  • NF-KappaB Inhibitor alpha
  • NF-kappa B / metabolism*
  • Oligonucleotide Array Sequence Analysis
  • Phosphorylation
  • Signal Transduction
  • Smad Proteins / metabolism*
  • Transforming Growth Factor beta / metabolism

Substances

  • Cytokines
  • Enzyme Inhibitors
  • I-kappa B Proteins
  • NF-kappa B
  • NFKBIA protein, human
  • Smad Proteins
  • Transforming Growth Factor beta
  • NF-KappaB Inhibitor alpha