Long-term benzodiazepine use and salivary cortisol: the Netherlands Study of Depression and Anxiety (NESDA)

J Clin Psychopharmacol. 2010 Apr;30(2):160-8. doi: 10.1097/JCP.0b013e3181d41f41.

Abstract

Background: As benzodiazepines (BZDs) have anxiolytic effects, it is expected that they influence the stress system. During short-term treatment, BZD use was found to suppress cortisol levels. However, little research has been done on the effects of long-term BZD administration on the hypothalamic-pituitary-adrenal (HPA) axis.

Methods: The association between long-term BZD use and cortisol levels was investigated in subjects of the Netherlands Study of Depression and Anxiety with a lifetime diagnosis of anxiety or depression (n = 1531). The subjects were categorized as "daily BZD users" (n = 96), "infrequent BZD users" (n = 172), and "nonusers" (n = 1263). Possible associations between characteristics of BZD use (dose, duration, and dependence) and salivary cortisol levels were analyzed.

Main outcome measure: Subjects provided 7 saliva samples, from which 4 cortisol indicators were calculated: the cortisol awakening response, diurnal slope, evening cortisol, and cortisol suppression after ingestion of 0.5 mg of dexamethasone.

Results: Daily users used BZDs for a median duration of 26.5 months and had a median daily dosage of 6.0 mg as measured in diazepam equivalents. Evening cortisol levels were significantly lower in daily users (P = 0.004; effect size: d = 0.24) and infrequent users (P = 0.04; effect size: d = 0.12) compared to nonusers. We did not find significant differences in the cortisol awakening response, diurnal slope, or in the dexamethasone suppression test.

Conclusions: Despite the finding of slightly lower evening cortisol levels in daily and infrequent BZD users compared to nonusers, results indicate that long-term BZD use is not convincingly associated with HPA axis alterations.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Anxiety Disorders / drug therapy
  • Anxiety Disorders / metabolism*
  • Anxiety Disorders / psychology
  • Benzodiazepines / administration & dosage*
  • Circadian Rhythm / drug effects
  • Circadian Rhythm / physiology
  • Cohort Studies
  • Cross-Sectional Studies
  • Depressive Disorder / drug therapy
  • Depressive Disorder / metabolism*
  • Depressive Disorder / psychology
  • Female
  • Humans
  • Hydrocortisone / chemistry
  • Hydrocortisone / metabolism*
  • Longitudinal Studies
  • Male
  • Middle Aged
  • Netherlands
  • Saliva / drug effects*
  • Saliva / metabolism*
  • Time Factors

Substances

  • Benzodiazepines
  • Hydrocortisone